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Search Results for " Angiotensin Receptor "

ターゲット

164

阻害剤

8

天然化合物

22

リコンビナントタンパク質

1

ライブラリー

カタログ番号 製品名 別名 ターゲット
TP1528 Angiotensin I/II (1-5) Angiotensin I/II 1-5 RAAS , Others
Angiotensin I/II (1-5) is a peptide (ASP-ARG-VAL-TYR-ILE) that contains the amino acids 1-5 and is converted from Angiotensin I/II.
TP1579 Angiotensin I/II (1-6) Angiotensin I/II 1-6 RAAS , Others
Angiotensin I/II (1-6) is a peptide (ASP-ARG-VAL-TYR-ILE-HIS) that contains the amino acids 1-6 and is converted from Angiotensin I/II peptide.
T7577 Angiotensin III, human, mouse Angiotensin III, human, mouse(3TFA) RAAS
Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA))(3TFA) is an endogenous angiotensin II receptor (AT2R) agonist(IC50s of 0.648 nM).
T7339 Angiotensin (1-7) Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO RAAS , Endogenous Metabolite
Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) is a synthetic heptapeptide identical to endogenous angiotensin-(1-7) , inhibits purified canine ACE activity (IC50=0.65 μM) with vasodilator and antiproliferative activiti...
T8560 Angiotensin II human acetate Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate Apoptosis , RAAS
Angiotensin II human acetate (DRVYIHPF acetate) is a vasoconstrictor that mainly acts on the AT1 receptor.
TP1929L1 Saralasin acetate(34273-10-4 free base) RAAS
Saralasin acetate is a Non-selective angiotensin II antagonist.
T3178 BIBS 39 RAAS
BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.
T2531 Eprosartan Mesylate SKF-108566J RAAS
Eprosartan Mesylate (SKF-108566J) is a competitive and reversible Angiotensin II Receptor Blocker.
T7354 H-Val-Pro-Pro-OH RAAS
H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).
T1461 Candesartan CV 11974 RAAS
Candesartan (CV 11974) is an angiotensin II receptor blocker used widely in the therapy of hypertension and heart failure.
T22344 Icatibant Acetate Bradykinin Receptor
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.
T13376 YS-49 RAAS , Akt , PI3K , Adrenergic Receptor
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T5355 Sparsentan RE-021,DARA-a RAAS , Endothelin Receptor
Sparsentan (DARA-a) is a first-in-class orally active and highly potent dual endothelin A and angiotensin II receptor antagonist(Ki of 9.3 and 0.8 nM, respectively)
T6067 PD 123319 (S)-(+)-PD 123319,PD123319 RAAS
PD 123319 ((S)-(+)-PD 123319) is a potent, selective AT2 angiotensin II receptor antagonist.
T1570 Telmisartan BIBR 277 RAAS , Autophagy
Telmisartan (BIBR 277) is an Angiotensin 2 Receptor Blocker. The mechanism of action of telmisartan is as an Angiotensin 2 Receptor Antagonist.
T0215L Losartan DuP-753 RAAS
Losartan (DuP-753) is an angiotensin II receptor antagonist.
T7797 Tasosartan WAY-ANA 756 RAAS
Tasosartan (WAY-ANA 756) is an antagonist of angiotensin II type 2 (AT2) receptor (IC50 = 1.2 nM).
T6219 Azilsartan Medoxomil TAK-491 RAAS
Azilsartan Medoxomil (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.
T3461 Losartan Carboxylic Acid EXP-3174,E-3174 RAAS
Losartan Carboxylic Acid (E-3174) a potent AT1 antagonist (Kis: 0.57 nM, rat; 0.67 nM, human), producing a depressor response and vasodilatation. Losartan Carboxylic Acid , a metabolite of losartan, is more potent than l...
T2318 Sacubitril/Valsartan Sacubitril mixture with Valsartan,Valsartan,Sacubitril,LCZ696 Apoptosis , RAAS , Neprilysin
Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for the treatment of hypertension and heart failure.
T1518 Olmesartan Medoxomil CS 866,Benicar RAAS
Olmesartan Medoxomil (Benicar) is an angiotensin II type 1 receptor blocker that is used to manage hypertension.
T2322 Fimasartan BR-A-657,Kanarb Apoptosis , RAAS
Fimasartan (BR-A-657) is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Concurrent administration of fimasartan with diuretic hydrochlorothiazide has show...
T4431 Olodanrigan PD-126055,EMA401 RAAS
Olodanrigan (EMA401), a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hyperexcitability and sprouting of DRG neurons. EMA...
T5964 Olmesartan CS 088,RNH 6270 RAAS
Olmesartan (RNH 6270) is an Angiotensin II Type I receptor antagonist. Olmesartan is the active form of the antihypertensive drug olmesartan medoxomil,and has antihypertensive activity.
T2270 Trans-Tranilast Tranilast trans- RAAS
Trans-Tranilast is an antiallergic drug developed by Kissei Pharmaceuticals. It was approved in 1982 for use in Japan and South Korea for bronchial asthma. Indications for keloid and hypertrophic scar were added in 1993....
T2400 Candesartan Cilexetil TCV-116 Apoptosis , RAAS
Candesartan Cilexetil (TCV-116) is an angiotensin II receptor antagonist (IC50: 0.26 nM). After hydrolysis of candesartan cilexetil to candesartan during gastrointestinal absorption, candesartan selectively competes with...
T5824 Angiotensin II (3-8), human Angiotensin IV RAAS
Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.
T6716 Valsartan Diovan,Tareg,CGP 48933 RAAS
Valsartan (CGP 48933) is a tetrazole derivative and angiotensin II type 1 receptor blocker that is used to treat hypertension.
T7575 [Sar1, Ile8]-Angiotensin II [Sar1, Ile8]-Angiotensin II(3TFA) RAAS , Others
[Sar1, Ile8]-Angiotensin II(3TFA) is a peptide that has multiple effects on vascular smooth muscle.
T1057 Azilsartan TAK-536 RAAS
Azilsartan (TAK-536) is an Angiotensin 2 Receptor Blocker. The mechanism of action of azilsartan is as an Angiotensin 2 Type 1 Receptor Antagonist. The physiologic effect of azilsartan is by means of Decreased Blood Pres...
T2690 Tranilast MK 341,SB 252218 RAAS , Prostaglandin Receptor
Tranilast (SB 252218), an antiallergic drug, suppresses lipid mediator and cytokine release from inflammatory cells, therefore utilized in the treatment of allergic disorders.
T19930 Nitrosoglutathione S-Nitrosoglutathione,SNOG,Glutathione thionitrite,GSNO RAAS , NO Synthase
Nitrosoglutathione (GSNO) is an endogenous transnitrosation donor involved in S-nitrosation of a variety of cellular proteins. GSNO, an exogenous NO donor and substrate of rat alcohol dehydrogenase class III isoenzyme, i...
T1615 Irbesartan SR-47436,BMS-186295 Apoptosis , RAAS
Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.
T0215 Losartan potassium DuP-753 potassium,MK 954,DuP 753 RAAS
Losartan potassium (DuP-753 potassium) , an Angiotensin II Receptor Blocker, selectively and competitively blocks the binding of angiotensin II to the angiotensin I (AT1) receptor.
T7616 A 779 RAAS
A 779 is a potent antagonist of the G-protein-coupled receptor Mas, the Ang1-7 receptor, which is distinct from conventional AngII.
TP1017L Angiotensin II 5-valine TFA Angiotensin II 5-valine TFA(58-49-1 free base) RAAS
Angiotensin II 5-valine TFA is an agonist of angiotensin receptor.
T13390 ZD 7155 hydrochloride RAAS
ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.
T7743 ANGIOTENSIN IV TFA(12676-15-2(free base)) RAAS
ANGIOTENSIN IV TFA is a less effective agonist at the angiotensin AT1 receptor.
T28540 Ripisartan UP 269-6,UP-2696,UP 2696,UP-269-6,UP269-6 RAAS
Ripisartan (UP-269-6) is a potent and specific angiotensin II receptor antagonist that inhibits angiotensin II-mediated sympathetic tachycardia responses.
T40220L TRV055 acetate TRV055 acetate (25849-90-5 Free base) RAAS
TRV055 acetate is a ligand of angiotensin II type 1 receptor and stimulates cellular Gq-mediated signaling.
T14942 CGP48369 RAAS
CGP48369 is a potent angiotensin II receptor antagonist with antihypertensive effects that enhances endothelium-dependent relaxation of coronary arteries in spontaneously hypertensive rats.
T14337 Buloxibutid AT2 receptor agonist C21 RAAS
Buloxibutid (AT2 receptor agonist C21) is a novel and selective small molecule angiotensin II AT2 receptor agonist with Ki values of 0.4 nM and 10 μM for AT2 and AT1 receptors, respectively.
T24588 Palatrigine BW-A 256C,BW A256C Adrenergic Receptor , Angiotensin-converting Enzyme (ACE)
Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.
T7616L A 779 TFA(159432-28-7 free base) A 779 3TFA(159432-28-7(free base)) RAAS
A 779 TFA is a potent antagonist of angiotensin-(1-7) receptor.
T67848 Valsartan Methyl Ester RAAS
Valsartan Methyl Ester is a potent angiotensin II receptor antagonist, IC50= 0.06uM.
T35834L (Sar¹)-Angiotensin II acetate RAAS
(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor. It binds to brain membrane-rich particles, with a Kd of 2.7 nM. It can stimulate protein synthesis and cell...
T27762 L-162,313 L-162313,L 162,313,L162,313 RAAS
L-162,313 is an ANG II receptor agonist, a nonpeptide that mimics the biological actions of angiotensin II and induces an increase in MAP.
T28437 Pomisartan BIBR-363,BIBR 363,BIBR363 RAAS
Pomisartan (BIBR-363) is a small molecule angiotensin type 1 receptor (AT1R) antagonist that is used in the treatment of cardiovascular disease, studying heart failure and hypertensio
T2531L Eprosartan KF-108566J free base,Teveten RAAS
Eprosartan (SKF-108566J free base) is a selective and competitive nonpeptide angiotensin II receptor antagonist with high affinity for AT1 receptor subtypes and can be used as an antihypertensive agent.Eprosartan has an ...
T65740 Trityl candesartan
Trityl candesartan is a crucial intermediate used in the synthesis of Candesartan and Candesartan cilexetil, which are angiotensin II receptor antagonists.

Compounds

Angiotensin I/II (1-5)
TP1528
Synonym: Angiotensin I/II 1-5
Target: RAAS, Others
Angiotensin I/II (1-6)
TP1579
Synonym: Angiotensin I/II 1-6
Target: RAAS, Others
Angiotensin III, human, mouse
T7577
Synonym: Angiotensin III, human, mouse(3TFA)
Target: RAAS
Angiotensin (1-7)
T7339
Synonym: Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO
Target: RAAS, Endogenous Metabolite
Angiotensin II human acetate
T8560
Synonym: Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate
Target: Apoptosis, RAAS
Saralasin acetate(34273-10-4 free base)
TP1929L1
Synonym:
Target: RAAS
BIBS 39
T3178
Synonym:
Target: RAAS
Eprosartan Mesylate
T2531
Synonym: SKF-108566J
Target: RAAS
H-Val-Pro-Pro-OH
T7354
Synonym:
Target: RAAS
Candesartan
T1461
Synonym: CV 11974
Target: RAAS
Icatibant Acetate
T22344
Synonym:
Target: Bradykinin Receptor
YS-49
T13376
Synonym:
Target: RAAS, Akt, PI3K, Adrenergic Receptor
Sparsentan
T5355
Synonym: RE-021,DARA-a
Target: RAAS, Endothelin Receptor
PD 123319
T6067
Synonym: (S)-(+)-PD 123319,PD123319
Target: RAAS
Telmisartan
T1570
Synonym: BIBR 277
Target: RAAS, Autophagy
Losartan
T0215L
Synonym: DuP-753
Target: RAAS
Tasosartan
T7797
Synonym: WAY-ANA 756
Target: RAAS
Azilsartan Medoxomil
T6219
Synonym: TAK-491
Target: RAAS
Losartan Carboxylic Acid
T3461
Synonym: EXP-3174,E-3174
Target: RAAS
Sacubitril/Valsartan
T2318
Synonym: Sacubitril mixture with Valsartan,Valsartan,Sacubitril,LCZ696
Target: Apoptosis, RAAS, Neprilysin
Olmesartan Medoxomil
T1518
Synonym: CS 866,Benicar
Target: RAAS
Fimasartan
T2322
Synonym: BR-A-657,Kanarb
Target: Apoptosis, RAAS
Olodanrigan
T4431
Synonym: PD-126055,EMA401
Target: RAAS
Olmesartan
T5964
Synonym: CS 088,RNH 6270
Target: RAAS
Trans-Tranilast
T2270
Synonym: Tranilast trans-
Target: RAAS
Candesartan Cilexetil
T2400
Synonym: TCV-116
Target: Apoptosis, RAAS
Angiotensin II (3-8), human
T5824
Synonym: Angiotensin IV
Target: RAAS
Valsartan
T6716
Synonym: Diovan,Tareg,CGP 48933
Target: RAAS
[Sar1, Ile8]-Angiotensin II
T7575
Synonym: [Sar1, Ile8]-Angiotensin II(3TFA)
Target: RAAS, Others
Azilsartan
T1057
Synonym: TAK-536
Target: RAAS
Tranilast
T2690
Synonym: MK 341,SB 252218
Target: RAAS, Prostaglandin Receptor
Nitrosoglutathione
T19930
Synonym: S-Nitrosoglutathione,SNOG,Glutathione thionitrite,GSNO
Target: RAAS, NO Synthase
Irbesartan
T1615
Synonym: SR-47436,BMS-186295
Target: Apoptosis, RAAS
Losartan potassium
T0215
Synonym: DuP-753 potassium,MK 954,DuP 753
Target: RAAS
A 779
T7616
Synonym:
Target: RAAS
Angiotensin II 5-valine TFA
TP1017L
Synonym: Angiotensin II 5-valine TFA(58-49-1 free base)
Target: RAAS
ZD 7155 hydrochloride
T13390
Synonym:
Target: RAAS
ANGIOTENSIN IV TFA(12676-15-2(free base))
T7743
Synonym:
Target: RAAS
Ripisartan
T28540
Synonym: UP 269-6,UP-2696,UP 2696,UP-269-6,UP269-6
Target: RAAS
TRV055 acetate
T40220L
Synonym: TRV055 acetate (25849-90-5 Free base)
Target: RAAS
CGP48369
T14942
Synonym:
Target: RAAS
Buloxibutid
T14337
Synonym: AT2 receptor agonist C21
Target: RAAS
Palatrigine
T24588
Synonym: BW-A 256C,BW A256C
Target: Adrenergic Receptor, Angiotensin-converting Enzyme (ACE)
A 779 TFA(159432-28-7 free base)
T7616L
Synonym: A 779 3TFA(159432-28-7(free base))
Target: RAAS
Valsartan Methyl Ester
T67848
Synonym:
Target: RAAS
(Sar¹)-Angiotensin II acetate
T35834L
Synonym:
Target: RAAS
L-162,313
T27762
Synonym: L-162313,L 162,313,L162,313
Target: RAAS
Pomisartan
T28437
Synonym: BIBR-363,BIBR 363,BIBR363
Target: RAAS
Eprosartan
T2531L
Synonym: KF-108566J free base,Teveten
Target: RAAS
Trityl candesartan
T65740
Synonym:
Target:
1 2 3 4
カタログ番号 製品名 別名 ターゲット
T7040 Angiotensin II human DRVYIHPF,Angiotensin II,Hypertensin II,Ang II Apoptosis , RAAS
Angiotensin II human (Ang II) is a biologically active peptide, a vasoconstrictor. Angiotensin II interacts with AT1R and AT2R to regulate blood pressure, stimulate sympathetic nerves, and increase aldosterone biosynthes...
T5S0106 Peimisine Ebeiensine RAAS , AChR
1. Peimisine (Ebeiensine) can affect M-receptor, excit β-receptor, restrain the release of internal calcium, and promote to releaseing nitrogen monoxidum in order to relax tracheal smooth muscle and relieve asthma. 2. Pe...
T2836 Isorhamnetin 3-methylquercetin,3'-Methylquercetin,Isorhamnetol,3'-Methoxyquercetin MEK , PI3K , Endogenous Metabolite
Isorhamnetin (3-methylquercetin) is the methylated metabolite of quercetin. Quercetin is an important dietary flavonoid with in vitro antioxidant activity. Isorhamnetin prevents endothelial cell injuries from oxidized LD...
T37298 Spinacine Endogenous Metabolite
Spinacine has been isolated from spinach and the roots of Panax ginseng. This conformationally constrained amino acid is a structural element in certain biologically active compounds as glucagon antagonists and angiotens...
T38593 1-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone
Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone9, a quinolone alkaloid derived from Evodia rutaecarpa, is a potent antagonist of the angiotensin II receptor, displaying an IC50 value of 48.2 μM.
TN4860 Pueroside B COX , PPAR
Pueroside B may can treat coronary heart disease, it can interact with two or more targets[peroxisome proliferator activated receptor γ (PPAR-γ), angiotensin-converting enzyme (ACE), hydroxymethylglutaryl coenzyme A rece...
TN1061 Ganoderol B Androgen Receptor
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate cancer and benign prostatic hyperplasia (BPH) therapy throu...
T75697 1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone, a diacylglycerol acyltransferase inhibitor and angiotensin II receptor blocker, exhibits IC50 values of 20.1 μM and 34.1 μM, respectively. Additionally, it demonstr...

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPH-02268 AGTR2 Protein, Human, Recombinant (His & SUMO) Human E. coli
Receptor for angiotensin II. Cooperates with MTUS1 to inhibit ERK2 activation and cell proliferation.
TMPH-02267 AGTRAP Protein, Human, Recombinant (His & Myc & SUMO) Human E. coli
Appears to be a negative regulator of type-1 angiotensin II receptor-mediated signaling by regulating receptor internalization as well as mechanism of receptor desensitization such as phosphorylation. Induces also a decr...
TMPY-02869 MMP-12 Protein, Human, Recombinant (catalytic domain) Human E. coli
Matrix metalloproteinases (MMPs) are a family of zinc-dependent endopeptidases that degrade components of the extracellular matrix (ECM) and play essential roles in various physiological processes such as morphogenesis, ...
TMPK-00913 SARS Spike S1 Protein (His & Avi), Biotinylated SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00439 SARS-COV-2 Spike RBD Protein (His & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00433 SARS-COV-2 Spike S1 Protein (hFc & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00434 SARS-COV-2 Spike RBD Protein (hFc & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00908 SARS Spike S1 Protein (hFc & Avi) SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00438 SARS-COV-2 Spike S Trimer Protein (His & Avi) SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00444 SARS-COV-2 Spike S1 NTD Protein (His & Flag) SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00911 SARS Spike RBD Protein (His & Avi) SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00440 SARS-COV-2 Spike S1 Protein (His & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00437 SARS-COV-2 Spike RBD Protein (His & Avi) SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00909 SARS Spike S1 Protein (hFc & Avi), Biotinylated SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00912 SARS Spike RBD Protein (His & Avi), Biotinylated SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00910 SARS Spike S1 Protein (His & Avi) SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00432 SARS-COV-2 Spike S1 Protein (hFc & Avi) SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00443 SARS-COV-2 (Omicron B.1.1.529) Spike S1 Protein (His & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00442 SARS-COV-2 (Omicron B.1.1.529) Spike S Trimer Protein (His & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPK-00441 SARS-COV-2 Spike S Trimer Protein (His & Avi), Biotinylated SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays k...
TMPY-06885 SARS-CoV-2 XBB.1.16 (Omicron) Spike S1+S2 trimer Protein (ECD, His)
The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4;...
TMPH-02274 JAK2 Protein, Human, Recombinant (His) Human E. coli
Non-receptor tyrosine kinase involved in various processes such as cell growth, development, differentiation or histone modifications. Mediates essential signaling events in both innate and adaptive immunity. In the cyto...
AGTR2 Protein, Human, Recombinant (His & SUMO)
TMPH-02268
Species: Human
Expression System: E. coli
AGTRAP Protein, Human, Recombinant (His & Myc & SUMO)
TMPH-02267
Species: Human
Expression System: E. coli
MMP-12 Protein, Human, Recombinant (catalytic domain)
TMPY-02869
Species: Human
Expression System: E. coli
SARS Spike S1 Protein (His & Avi), Biotinylated
TMPK-00913
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (His & Avi), Biotinylated
TMPK-00439
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (hFc & Avi), Biotinylated
TMPK-00433
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (hFc & Avi), Biotinylated
TMPK-00434
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike S1 Protein (hFc & Avi)
TMPK-00908
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike S Trimer Protein (His & Avi)
TMPK-00438
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 NTD Protein (His & Flag)
TMPK-00444
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike RBD Protein (His & Avi)
TMPK-00911
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (His & Avi), Biotinylated
TMPK-00440
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (His & Avi)
TMPK-00437
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike S1 Protein (hFc & Avi), Biotinylated
TMPK-00909
Species: SARS
Expression System: HEK293 Cells
SARS Spike RBD Protein (His & Avi), Biotinylated
TMPK-00912
Species: SARS
Expression System: HEK293 Cells
SARS Spike S1 Protein (His & Avi)
TMPK-00910
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (hFc & Avi)
TMPK-00432
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 (Omicron B.1.1.529) Spike S1 Protein (His & Avi), Biotinylated
TMPK-00443
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 (Omicron B.1.1.529) Spike S Trimer Protein (His & Avi), Biotinylated
TMPK-00442
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S Trimer Protein (His & Avi), Biotinylated
TMPK-00441
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 XBB.1.16 (Omicron) Spike S1+S2 trimer Protein (ECD, His)
TMPY-06885
Species:
Expression System:
JAK2 Protein, Human, Recombinant (His)
TMPH-02274
Species: Human
Expression System: E. coli
カタログ番号 製品名
L7110 Anti-Hypertension Compound Library

678 compounds
678 hypertension-related small molecules for high-throughput and high-content screening.